Search results for "S. aureu"

showing 10 items of 10 documents

Synthesis and biofilm formation reduction of pyrazole-4-carboxamide derivatives in some Staphylococcus aureus strains

2016

The ability of several N-phenyl-1H-pyrazole-4-carboxamide derivatives and other pyrazoles opportunely modified at the positions 3, 4 and 5, to reduce the formation of the biofilm in some Staphylococcus aureus strains (ATCC 29213, ATCC 25923 and ATCC 6538) were investigated. All the tested compounds were able, although to a different extent, to reduce the biofilm formation of the three bacterial strains considered. Among these, the 1-(2,5-dichlorophenyl)-5-methyl-N-phenyl-1H-pyrazole-4-carboxamide 14 resulted as the best inhibitor of biofilm formation showing an IC50 ranging from 2.3 to 32 μM, against all the three strains of S. aureus. Compound 14 also shows a good protective effect in vivo…

0301 basic medicineStaphylococcus aureusmedicine.drug_class030106 microbiologyCarboxamideMothsN-phenyl-1H-pyrazole-4-carboxamidePyrazoleSettore BIO/19 - Microbiologia Generalemedicine.disease_cause01 natural sciencesMicrobiologyStructure-Activity Relationship03 medical and health scienceschemistry.chemical_compoundDrug DiscoveryInhibition of biofilm formationmedicineAnimalsIC50PharmacologyWaxVirulencebiology010405 organic chemistryDrug Discovery3003 Pharmaceutical ScienceAnti-virulenceOrganic ChemistryBiofilmS. aureuGeneral MedicineStaphylococcal Infectionsbiology.organism_classificationSettore CHIM/08 - Chimica FarmaceuticaAnti-Bacterial Agents0104 chemical sciencesGalleria mellonellaHydrazinesSettore AGR/11 - Entomologia Generale E ApplicatachemistryStaphylococcus aureusBiofilmsLarvavisual_artWax moth larva modelvisual_art.visual_art_mediumPyrazolesLead compoundEuropean Journal of Medicinal Chemistry
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Metabolic Adaptation and Protein Complexes in Prokaryotes.

2012

Protein complexes are classified and have been charted in several large-scale screening studies in prokaryotes. These complexes are organized in a factory-like fashion to optimize protein production and metabolism. Central components are conserved between different prokaryotes; major complexes involve carbohydrate, amino acid, fatty acid and nucleotide metabolism. Metabolic adaptation changes protein complexes according to environmental conditions. Protein modification depends on specific modifying enzymes. Proteins such as trigger enzymes display condition-dependent adaptation to different functions by participating in several complexes. Several bacterial pathogens adapt rapidly to intrace…

Endocrinology Diabetes and MetabolismMetaboliteSubstrate channelinglcsh:QR1-502ReviewBiologyBiochemistrylcsh:Microbiologyprokaryoteschemistry.chemical_compoundDownregulation and upregulationGene expressionProtein biosynthesisMolecular Biologymetaboliteschemistry.chemical_classificationprotein complexesE. coliMetabolismS. aureuschannelingAmino acidcrowdingEnzymechemistryBiochemistry
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Portraying infective endocarditis

2019

Infective endocarditis is a growing problem with many shifts due to ever-increasing comorbid illnesses, invasive procedures, and increase in the elderly. We performed this multinational study to depict definite infective endocarditis. Adult patients with definite endocarditis hospitalized between January 1, 2015, and October 1, 2018, were included from 41 hospitals in 13 countries. We included microbiological features, types and severity of the disease, complications, but excluded therapeutic parameters. A total of 867 patients were included. A total of 631 (72.8%) patients had native valve endocarditis (NVE), 214 (24.7%) patients had prosthetic valve endocarditis (PVE), 21 (2.4%) patients …

MaleInternationalityAucunInfective endocarditimedicine.disease_causeMedical microbiology80 and overBlood cultureHospital MortalityAged 80 and overmedicine.diagnostic_testbiologyEndocarditisSBacterialGeneral MedicineSciences bio-médicales et agricolesMiddle AgedStaphylococcal InfectionsSciences du Vivant [q-bio]/Microbiologie et ParasitologieViridans StreptococciCatheterInfectious Diseases[SDV.MP]Life Sciences [q-bio]/Microbiology and ParasitologyStaphylococcus aureusInfective endocarditisAortic ValveMitral ValveFemaleMicrobiology (medical)Adultmedicine.medical_specialtyProsthesis-Related InfectionsAdolescentaureusBlood cultureYoung AdultInternal medicinemedicineEndocarditisHumansresults of multinational ID-IRI study- EUROPEAN JOURNAL OF CLINICAL MICROBIOLOGY & INFECTIOUS DISEASES cilt.38 ss.1753-1763 2019 [Erdem H. Puca E. Ruch Y. Santos L. Ghanem-Zoubi N. Argemi X. Hansmann Y. Guner R. Tonziello G. Mazzucotelli J. et al. -Portraying infective endocarditis]ProstheticAgedNative Valve EndocarditisBacteriabusiness.industryEndocarditis Bacterialmedicine.diseasebiology.organism_classificationS. aureusViridans streptococciInfective endocarditisbusinessNative
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Application of fnbA gene as new target for the species-specific and quantitative detection of Staphylococcus aureus directly from lower respiratory t…

2013

Staphylococcus aureus is a significant cause of hospital-acquired pneumonia (HAP), particularly in mechanically ventilated patients. We used the fibronectin-binding protein A gene (fnbA) for the species-specific and quantitative detection of S. aureus directly from lower respiratory tract (LRT) specimens by a Taq Man real time PCR. For this reason, a total of 269 lower respiratory tract (LRT) specimens collected from patients with hospital-acquired pneumonia were assayed. Amplification of fnbA in serial dilutions ranged from 10(9) CFU/ ml to 10(2) CFU/ml. Standard curve of triplicate every dilution had slope 3.34±0.1 and R2>0.99 with SD 0.1. Based on these data, the sensitivity and specif…

Microbiology (medical)fnbA Gene real time PCR respiratory infection Staphylococcus aureusSettore MED/07 - Microbiologia E Microbiologia ClinicaStaphylococcus aureusSerial dilutionRespiratory Systemlcsh:QR1-502medicine.disease_causeReal-Time Polymerase Chain ReactionSensitivity and SpecificityfnbA Genelcsh:MicrobiologyPathology and Forensic MedicineMicrobiologyrespiratory infectionPneumonia StaphylococcalmedicineTaqManlcsh:PathologyHumansAdhesins BacterialCross InfectionbiologyStaphylococcus. aureusRespiratory infectionGeneral Medicinemedicine.diseasePneumoniareal time PCRmedicine.anatomical_structureReal-time polymerase chain reactionMolecular Diagnostic TechniquesStaphylococcus aureusbiology.proteinProtein ARespiratory tractlcsh:RB1-214Indian journal of pathologymicrobiology
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Propolis-Based Nanofiber Patches to Repair Corneal Microbial Keratitis

2021

In this research, polyvinyl-alcohol (PVA)/gelatin (GEL)/propolis (Ps) biocompatible nanofiber patches were fabricated via electrospinning technique. The controlled release of Propolis, surface wettability behaviors, antimicrobial activities against the S. aureus and P. aeruginosa, and biocompatibility properties with the mesenchymal stem cells (MSCs) were investigated in detail. By adding 0.5, 1, and 3 wt.% GEL into the 13 wt.% PVA, the morphological and mechanical results suggested that 13 wt.% PVA/0.5 wt.% GEL patch can be an ideal matrix for 3 and 5 wt.% propolis addition. Morphological results revealed that the diameters of the electrospun nanofiber patches were increased with GEL (from…

Pharmaceutical ScienceBiocompatible Materials02 engineering and technologyGelatinAnalytical ChemistryContact angleQD241-4410302 clinical medicineAnti-Infective AgentsSpectroscopy Fourier Transform InfraredDrug DiscoveryMesenchymal stem cell proliferationDrug CarriersChemistrySSCAFFOLDHYDROGELP<i>S. aureus</i>021001 nanoscience & nanotechnologyControlled releaseaeruginosaElectrospinningpropolisChemistry (miscellaneous)microbial keratitisPseudomonas aeruginosaBLINDNESSMolecular MedicineELECTROSPUN0210 nano-technologyStaphylococcus aureusfood.ingredient<i>P. aeruginosa</i>BiocompatibilitySurface PropertiesFABRICATIONMicrobial Sensitivity TestsCHEMICAL-COMPOSITIONaureusArticle03 medical and health sciencesfoodnanofibersPhysical and Theoretical Chemistrycorneal patchelectrospinningKeratitisCOMPOSITEGELATINOrganic ChemistryPropolisS. aureusDrug LiberationP. aeruginosaPolyvinyl AlcoholNanofiber030221 ophthalmology & optometryPROPERTYMEMBRANENuclear chemistry
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Straightforward Approach for Preparing Durable Antibacterial ZnO Nanoparticle Coatings on Flexible Substrates

2022

Flexible antibacterial materials have gained utmost importance in protection from the distribution of bacteria and viruses due to the exceptional variety of applications. Herein, we demonstrate a readily scalable and rapid single-step approach for producing durable ZnO nanoparticle antibacterial coating on flexible polymer substrates at room temperature. Substrates used are polystyrene, poly(ethylene-co-vinyl acetate) copolymer, poly(methyl methacrylate), polypropylene, high density polyethylene and a commercial acrylate type adhesive tape. The deposition was achieved by a spin-coating process using a slurry of ZnO nanoparticles in toluene. A stable modification layer was obtained when tolu…

PolymersnanoparticleOrganic ChemistryE. coliPharmaceutical Sciencecoating:NATURAL SCIENCES::Physics [Research Subject Categories]S. aureus540ZnO; nanoparticle; coating; flexible substrate; antibacterial; <i>E. coli</i>; <i>S. aureus</i>Anti-Bacterial AgentsAnalytical Chemistryantibacterialflexible substrateChemistry (miscellaneous)Drug DiscoveryEscherichia coliSolventsZnOPolystyrenesMolecular MedicineZinc OxidePhysical and Theoretical ChemistryToluene
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Lipid and phase specificity of α-toxin from S. aureus

2013

AbstractThe pore forming toxin Hla (α-toxin) from Staphylococcus aureus is an important pathogenic factor of the bacterium S. aureus and also a model system for the process of membrane-induced protein oligomerisation and pore formation. It has been shown that binding to lipid membranes at neutral or basic pH requires the presence of a phosphocholine-headgroup. Thus, sphingomyelin and phosphatidylcholine may serve as interaction partners in cellular membranes. Based on earlier studies it has been suggested that rafts of sphingomyelin are particularly efficient in toxin binding. In this study we compared the oligomerisation of Hla on liposomes of various lipid compositions in order to identif…

Staphylococcus aureusPore formationLiquid ordered phaseBacterial ToxinsLipid BilayersBiophysicsBiologyBiochemistryPhase Transitionchemistry.chemical_compoundHemolysin ProteinsMembrane LipidsMembrane MicrodomainsPhosphatidylcholineBinding siteLipid raftUnilamellar LiposomesPore-forming toxinLiposomeArtificial membranesBinding SitesCell MembraneOligomerisationCell BiologyS. aureusSphingomyelinsMembraneBiochemistrychemistryMicroscopy FluorescenceMutationPhosphatidylcholineslipids (amino acids peptides and proteins)Protein MultimerizationToxinSphingomyelinBiochimica et Biophysica Acta (BBA) - Biomembranes
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Cilvēka mikroflora kā potenciāls acs infekcijas avots

2015

Bakalaura darbs uzrakstīts latviešu valodā. Mērķis: novērtēt cilvēka normālās mikrofloras iespējamo lomu acu slimību etioloģijā un patoģenēzē. Uzdevumi: noteikt S.aureus nēsātāju izplatību sabiedrībā; novērtēt roku mazgāšanas un dezinfekcijas efektivitāti; noteikt no dezinficēto roku ādas izolēto KONS jutību pret antibiotikām. Metode: tika veikti mikrobioģiskie uzsējumi un izaugušo koloniju uzskaitījums. Paraugi iegūti no deguna un roku ādas. Uzņēmība pret 6 antibiotikām tika noteikta ar disku difūzijas metodi. Rezultāti: 1.16,96% dalībnieku ir pastāvīgi S.aureus nēsātāji degunā. 2.Efektīvākais pretmikrobu līdzeklis ir 96% medicīniskais spirts. 3.No dezinficēto roku ādas tika izolēti potenc…

antibakteriālā rezistenceFizikaS.epidermidisS. aureus
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eIF2α confers cellular tolerance to S. aureus α-toxin

2015

We report on the role of conserved stress-response pathways for cellular tolerance to a pore forming toxin. First, we observed that small molecular weight inhibitors including of eIF2α-phosphatase, jun-N-terminal kinase (JNK), and PI3-kinase sensitized normal mouse embryonal fibroblasts (MEFs) to the small pore forming S. aureus α-toxin. Sensitization depended on expression of mADAM10, the murine ortholog of a proposed high-affinity receptor for α-toxin in human cells. Similarly, eIF2α (S51A/S51A) MEFs, which harbor an Ala knock-in mutation at the regulated Ser51 phosphorylation site of eukaryotic translation initiation factor 2α, were hyper-sensitive to α-toxin. Inhibition of translation w…

lcsh:Immunologic diseases. AllergyMAPK/ERK pathwayImmunologyeIF2αBiologyCycloheximide03 medical and health scienceschemistry.chemical_compoundCellular toleranceImmunology and AllergyInitiation factorpore forming toxinsReceptorOriginal Research030304 developmental biologyGenetics0303 health sciencesKinase030302 biochemistry & molecular biologyJNK Mitogen-Activated Protein KinasesADAM10Translation (biology)MAPKCell biologyEIF2AK4chemistryPhosphorylationCytolysinS. aureus α-toxinlcsh:RC581-607Frontiers in Immunology
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Cytotoksyczność wybranych metaloftalocyjanin wobec mikroorganizmów

2015

Dokonano przeglądu literatury w zakresie cytotoksyczności metaloftalocyjanin wobec mikroorganizmów. W pracy zwrócono uwagę przede wszystkim na właściwości fotosensybilizacyjne ftalocyjanin oraz metaloftalocyjanin, które mogą być wykorzystane w terapii fotodynamicznej (PDT) oraz w fotodynamicznej terapii skierowanej przeciwko mikroorganizmom (PACT). Wykazano, że metalo-ftalocyjaniny bez podstawników, jak i kompleksy z podstawnikami aksjalnymi i/lub peryferyjnymi (t.j. pirydyna, grupy sulfonowe lub aminowe), a także ftalocyjaniny kationowe mogą być skuteczne w zwalczaniu bakterii (S. aureus E. coli), grzybów (np. S. cerevisiae) oraz wirusów (HSV). Działanie tych związków zależy głównie od moż…

metaloftalocyjaninyE. coliS. cerevisiaecytotoksycznośćS. aureus
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